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1

Mechanistic Studies on Metabolic Interactions between Gemfibrozil and Statins

Prueksaritanont, T.

Journal:

Journal of Pharmacology and Experimental Therapeutics

Année:

2002

Langue:

english

Fichier:

PDF, 239 KB

english, 2002

2

2,3-Diaminopyridine as a platform for designing structurally unique nonpeptide bradykinin B1 receptor antagonists

Dong-Mei Feng, Jenny M. Wai, Scott D. Kuduk, Christina Ng, Kathy L. Murphy, Richard W. Ransom, Duane Reiss, Raymond S.L. Chang, Charles M. Harrell, Tanya MacNeil, Cuyue Tang, Thomayant Prueksaritanont

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2005

Langue:

english

Fichier:

PDF, 112 KB

english, 2005

3

Bradykinin B1 antagonists: Biphenyl SAR studies in the cyclopropanecarboxamide series

Scott D. Kuduk, Robert M. DiPardo, Ronald K. Chang, Christina N. Di Marco, Kathy L. Murphy, Richard W. Ransom, Duane R. Reiss, Cuyue Tang, Thomayant Prueksaritanont, Douglas J. Pettibone, Mark G. Bock

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2007

Langue:

english

Fichier:

PDF, 148 KB

english, 2007

4

The human hepatic metabolism of simvastatin hydroxy acid is mediated primarily by CYP3A, and not CYP2D6

Thomayant Prueksaritanont, Bennett Ma, Nathan Yu

Journal:

British Journal of Clinical Pharmacology

Année:

2003

Langue:

english

Fichier:

PDF, 112 KB

english, 2003

5

Interconversion Pharmacokinetics of Simvastatin and its Hydroxy Acid in Dogs: Effects of Gemfibrozil

Thomayant Prueksaritanont, Yue Qiu, Lillian Mu, Kimberly Michel, Janice Brunner, Karen M. Richards, Jiunn H. Lin

Journal:

Pharmaceutical Research

Année:

2005

Langue:

english

Fichier:

PDF, 447 KB

english, 2005

6

An Extended Point-Area Deconvolution Approach for Assessing Drug Input Rates

Kuang C. Yeh, Daniel J. Holder, Gregory A. Winchell, Larissa A. Wenning, Thomayant Prueksaritanont

Journal:

Pharmaceutical Research

Année:

2001

Langue:

english

Fichier:

PDF, 197 KB

english, 2001

7

Impact of methionine oxidation on the binding of human IgG1 to FcRn and Fcγ receptors

Andrea Bertolotti-Ciarlet, Weirong Wang, Rebecca Lownes, Pavlo Pristatsky, Yulin Fang, Troy McKelvey, Yingzhe Li, Yunsong Li, James Drummond, Thomayant Prueksaritanont, Josef Vlasak

Journal:

Molecular Immunology

Année:

2009

Langue:

english

Fichier:

PDF, 499 KB

english, 2009

8

Drug–Drug Interaction Studies: Regulatory Guidance and An Industry Perspective

Prueksaritanont, Thomayant, Chu, Xiaoyan, Gibson, Christopher, Cui, Donghui, Yee, Ka Lai, Ballard, Jeanine, Cabalu, Tamara, Hochman, Jerome

Journal:

The AAPS Journal

Année:

2013

Langue:

english

Fichier:

PDF, 368 KB

english, 2013

9

Cyclopropylamino Acid Amide as a Pharmacophoric Replacement for 2,3-Diaminopyridine. Application to the Design of Novel Bradykinin B 1 Receptor Antagonists

Wood, Michael R., Schirripa, Kathy M., Kim, June J., Wan, Bang-Lin, Murphy, Kathy L., Ransom, Richard W., Chang, Raymond S. L., Tang, Cuyue, Prueksaritanont, Thomayant, Detwiler, Theodore J., Hettrick

Journal:

Journal of Medicinal Chemistry

Année:

2006

Langue:

english

Fichier:

PDF, 49 KB

english, 2006

10

Drug-Drug Interactions Related to Altered Absorption and Plasma Protein Binding: Theoretical and Regulatory Considerations, and an Industry Perspective

Hochman, Jerome, Tang, Cuyue, Prueksaritanont, Thomayant

Journal:

Journal of Pharmaceutical Sciences

Année:

2015

Langue:

english

Fichier:

PDF, 164 KB

english, 2015

11

Pharmacokinetic de-risking tools for selection of monoclonal antibody lead candidates

Dostalek, Miroslav, Prueksaritanont, Thomayant, Kelley, Robert F.

Journal:

Année:

2017

Langue:

english

Fichier:

PDF, 1.84 MB

english, 2017

12

Effects of pentobarbital on pharmacokinetics and pharmacodynamics of a potent fibrinogen receptor antagonist, L-734 217, in dogs

T. Prueksaritanont, M. T. Stranieri, E. L. Hand, J. D. Ellis, M. A. Holahan, G. R. Sitko, J. J. Cook

Journal:

Biopharmaceutics & Drug Disposition

Année:

1997

Langue:

english

Fichier:

PDF, 364 KB

english, 1997

13

Renal and non-renal clearances of iothalamate

Thomayant Prueksaritanont, Chung Y. Lui, Myung G. Lee, Win L. Chiou

Journal:

Biopharmaceutics & Drug Disposition

Année:

1986

Langue:

english

Fichier:

PDF, 438 KB

english, 1986

14

Absorption of iothalamate after oral administration and absorption enhancement by amino acids in dogs and rats

Thomayant Prueksaritanont, Myung G. Lee, Fung-Hwa Hsu, Win L. Chiou

Journal:

Biopharmaceutics & Drug Disposition

Année:

1986

Langue:

english

Fichier:

PDF, 773 KB

english, 1986

15

Absorption of iothalamate after oral administration: A preliminary study in humans and interspecies differences

Thomayant Prueksaritanont, Win L. Chiou

Journal:

Biopharmaceutics & Drug Disposition

Année:

1987

Langue:

english

Fichier:

PDF, 166 KB

english, 1987

16

Prediction of human clearance of therapeutic proteins: simple allometric scaling method revisited

Weirong Wang, Thomayant Prueksaritanont

Journal:

Biopharmaceutics & Drug Disposition

Année:

2010

Langue:

english

Fichier:

PDF, 127 KB

english, 2010

17

Nonpeptide αvβ3 Antagonists: Identification of Potent, Chain-Shortened 7-Oxo RGD Mimetics.

Amy E. Zartman, Le T. Duong, Carmen Fernandez-Metzler, George D. Hartman, Chih-Tai Leu, Thomayant Prueksaritanont, Gideon A. Rodan, Sevgi B. Rodan, Mark E. Duggan, Robert S. Meissner

Journal:

Année:

2005

Fichier:

PDF, 20 KB

2005

18

Using real-time quantitative TaqMan RT-PCR to evaluate the role of dexamethasone in gene regulation of rat P-glycoproteins mdr1a/1b and cytochrome P450 3A1/2

Qin Mei, Karen Richards, Kristie Strong-Basalyga, Scott E. Fauty, Anne Taylor, Masayo Yamazaki, Thomayant Prueksaritanont, Jiunn H. Lin, Jerome Hochman

Journal:

Journal of Pharmaceutical Sciences

Année:

2004

Langue:

english

Fichier:

PDF, 159 KB

english, 2004

19

Nonpeptide αvβ3 antagonists. Part 10: In vitro and in vivo evaluation of a potent 7-methyl substituted tetrahydro-[1,8]naphthyridine derivative

Michael J Breslin, Mark E Duggan, Wasyl Halczenko, George D Hartman, Le T Duong, Carmen Fernandez-Metzler, Michael A Gentile, Donald B Kimmel, Chih-Tai Leu, Kara Merkle, Thomayant Prueksaritanont, Gid

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2004

Langue:

english

Fichier:

PDF, 260 KB

english, 2004

20

Nonpeptide αvβ3 antagonists. Part 9: Improved pharmacokinetic profile through the use of an aliphatic, des-amide backbone

David B. Whitman, Ben C. Askew, Le T. Duong, Carmen Fernandez-Metzler, Wasyl Halczenko, George D. Hartman, John H. Hutchinson, Chih-Tai Leu, Thomayant Prueksaritanont, Gideon A. Rodan, Sevgi B. Rodan,

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2004

Langue:

english

Fichier:

PDF, 257 KB

english, 2004

21

Nonpeptide αvβ3 antagonists: identification of potent, chain-shortened 7-oxo RGD mimetics

Amy E. Zartman, Le T. Duong, Carmen Fernandez-Metzler, George D. Hartman, Chih-Tai Leu, Thomayant Prueksaritanont, Gideon A. Rodan, Sevgi B. Rodan, Mark E. Duggan, Robert S. Meissner

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2005

Langue:

english

Fichier:

PDF, 115 KB

english, 2005

22

Bradykinin B1 antagonists: SAR studies in the 2,3-diaminopyridine series

Scott D. Kuduk, Ronald K. Chang, Christina Ng, Kathy L. Murphy, Richard W. Ransom, Cuyue Tang, Thomayant Prueksaritanont, Roger M. Freidinger, Douglas J. Pettibone, Mark G. Bock

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2005

Langue:

english

Fichier:

PDF, 197 KB

english, 2005

23

A new class of bradykinin B1 receptor antagonists with high oral bioavailability and minimal PXR activity

Dong-Mei Feng, Robert M. DiPardo, Jenny M. Wai, Ronald K. Chang, Christina N. Di Marco, Kathy L. Murphy, Richard W. Ransom, Duane R. Reiss, Cuyue Tang, Thomayant Prueksaritanont, Douglas J. Pettibone,

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2008

Langue:

english

Fichier:

PDF, 154 KB

english, 2008

24

Bradykinin B1 receptor antagonists: An α-hydroxy amide with an improved metabolism profile

Scott D. Kuduk, Ronald K. Chang, Robert M. DiPardo, Christina N. Di Marco, Kathy L. Murphy, Richard W. Ransom, Duane R. Reiss, Cuyue Tang, Thomayant Prueksaritanont, Douglas J. Pettibone, Mark G. Bock

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2008

Langue:

english

Fichier:

PDF, 169 KB

english, 2008

25

Design and synthesis of conformationally constrained N,N-disubstituted 1,4-diazepanes as potent orexin receptor antagonists

Paul J. Coleman, John D. Schreier, Georgia B. McGaughey, Michael J. Bogusky, Christopher D. Cox, George D. Hartman, Richard G. Ball, C. Meacham Harrell, Duane R. Reiss, Thomayant Prueksaritanont, Chri

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 612 KB

english, 2010

26

Indazole derivatives as novel bradykinin B1 receptor antagonists

Vera Bodmer-Narkevitch, Neville J. Anthony, Victoria Cofre, Samson M. Jolly, Kathy L. Murphy, Richard W. Ransom, Duane R. Reiss, Cuyue Tang, Thomayant Prueksaritanont, Douglas J. Pettibone, Mark G. Bo

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 1.32 MB

english, 2010

27

Simple and micro high-performance liquid chromatographic method for simultaneous determination of p-aminohippuric acid and iothalamate in biological fluids

Thomayant Prueksaritanont, Mei-Ling Chen, Win L. Chiou

Journal:

Journal of Chromatography B: Biomedical Sciences and Applications

Année:

1984

Langue:

english

Fichier:

PDF, 589 KB

english, 1984

28

Simultaneous determination of ranitidine and its metabolites in human plasma and urine by high-performance liquid chromatography

Thomayant Prueksaritanont, Nantana Sittichai, Somjit Prueksaritanont, Rewadee Vongsaroj

Journal:

Journal of Chromatography B: Biomedical Sciences and Applications

Année:

1989

Langue:

english

Fichier:

PDF, 621 KB

english, 1989

29

Creatinine : XIII. Micro high-performance liquid chromatographic assay of creatinine in biological fluids using fixed- or variable-wavelength UV detector

Win L. Chiou, Francis S. Pu, Thomayant Prueksaritanont

Journal:

Journal of Chromatography B: Biomedical Sciences and Applications

Année:

1983

Langue:

english

Fichier:

PDF, 227 KB

english, 1983

30

Non-Peptide αvβ3 Antagonists. Part 4: Potent and Orally Bioavailable Chain-Shortened RGD Mimetics

Paul J. Coleman, Ben C. Askew, John H. Hutchinson, David B. Whitman, James J. Perkins, George D. Hartman, Gideon A. Rodan, Chih-Tai Leu, Thomayant Prueksaritanont, Carmen Fernandez-Metzler, Kara M. Me

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2002

Langue:

english

Fichier:

PDF, 114 KB

english, 2002

31

Non-peptide αvβ3 antagonists. Part 5: identification of potent RGD mimetics incorporating 2-aryl β-amino acids as aspartic acid replacements

Karen M Brashear, Cecilia A Hunt, Brian T Kucer, Mark E Duggan, George D Hartman, Gideon A Rodan, Sevgi B Rodan, Chi-Tai Leu, Thomayant Prueksaritanont, Carmen Fernandez-Metzler, Andrea Barrish, Carl

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2002

Langue:

english

Fichier:

PDF, 120 KB

english, 2002

32

Metabolic interactions between mibefradil and HMG-CoA reductase inhibitors: an in vitro investigation with human liver preparations

Thomayant Prueksaritanont, Bennett Ma, Cuyue Tang, Yuan Meng, Carol Assang, Ping Lu, Paul J. Reider, Jiunn H. Lin, Thomas A. Baillie

Journal:

British Journal of Clinical Pharmacology

Année:

1999

Langue:

english

Fichier:

PDF, 136 KB

english, 1999

33

Comparative Effects of Fibrates on Drug Metabolizing Enzymes in Human Hepatocytes

Thomayant Prueksaritanont, Karen M. Richards, Yue Qiu, Kristine Strong-Basalyga, Alisha Miller, Chunze Li, Roy Eisenhandler, Edward J. Carlini

Journal:

Pharmaceutical Research

Année:

2005

Langue:

english

Fichier:

PDF, 298 KB

english, 2005

34

Use ofIn VivoAnimal Models to Assess Pharmacokinetic Drug-Drug Interactions

Cuyue Tang, Thomayant Prueksaritanont

Journal:

Pharmaceutical Research

Année:

2010

Langue:

english

Fichier:

PDF, 304 KB

english, 2010

35

Theoretical Analysis of Interplay of Therapeutic Protein Drug and Circulating Soluble Target: Temporal Profiles of ‘Free’ and ‘Total’ Drug and Target

Cuyue Tang, Thomayant Prueksaritanont

Journal:

Pharmaceutical Research

Année:

2011

Langue:

english

Fichier:

PDF, 523 KB

english, 2011

36

Non-peptide αvβ3 antagonists: Identification of potent, chain-shortened RGD mimetics that incorporate a central pyrrolidinone constraint

James J Perkins, L.T Duong, Carmen Fernandez-Metzler, George D Hartman, Donald B Kimmel, Chih-Tai Leu, Joseph J Lynch, Thomayant Prueksaritanont, Gideon A Rodan, Sevgi B Rodan, Mark E Duggan, Robert S

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2003

Langue:

english

Fichier:

PDF, 143 KB

english, 2003

37

Analysis of metabolite kinetics by deconvolution and in vivo–in vitro correlations of metabolite formation rates: Studies of fibrinogen receptor antagonist ester prodrugs

Thomayant Prueksaritanont, Lynn M. Gorham, Kuang C. Yeh

Journal:

Journal of Pharmaceutical Sciences

Année:

1997

Langue:

english

Fichier:

PDF, 157 KB

english, 1997

38

Bioavailability of cyclosporine with concomitant rifampin administration is markedly less than predicted by hepatic enzyme induction

Hebert, Mary F, Roberts, John P, Prueksaritanont, Thomayant, Benet, Leslie Z

Journal:

Clinical Pharmacology & Therapeutics

Année:

1992

Langue:

english

Fichier:

PDF, 698 KB

english, 1992

39

HPLC Assay for FK 506 and Two Metabolites in Isolated Rat Hepatocytes and Rat Liver Microsomes

Beatrice Y. T. Perotti, Thomayant Prueksaritanont, Leslie Z. Benet

Journal:

Pharmaceutical Research

Année:

1994

Fichier:

PDF, 690 KB

1994

40

Interactions of Human P-glycoprotein with Simvastatin, Simvastatin Acid, and Atorvastatin

Jerome H. Hochman, Nicole Pudvah, Julia Qiu, Masayo Yamazaki, Cuyue Tang, Jiunn H. Lin, Thomayant Prueksaritanont

Journal:

Pharmaceutical Research

Année:

2004

Langue:

english

Fichier:

PDF, 119 KB

english, 2004

41

Monoclonal Antibodies with Identical Fc Sequences Can Bind to FcRn Differentially with Pharmacokinetic Consequences

Wang, W., Lu, P., Fang, Y., Hamuro, L., Pittman, T., Carr, B., Hochman, J., Prueksaritanont, T.

Journal:

Drug Metabolism and Disposition

Année:

2011

Langue:

english

Fichier:

PDF, 1.12 MB

english, 2011

42

Non-Peptide αvβ3 antagonists. Part 6: Design and synthesis of αvβ3 antagonists containing a pyridone or pyrazinone central scaffold

Michael J Breslin, Mark E Duggan, Wasyl Halczenko, Carmen Fernandez-Metzler, Cecilia A Hunt, Chih-Tai Leu, Kara M Merkle, Adel M Naylor-Olsen, Thomayant Prueksaritanont, Gary Stump, Audrey Wallace, Se

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2003

Langue:

english

Fichier:

PDF, 192 KB

english, 2003

43

Effects of Fibrates on Metabolism of Statins in Human Hepatocytes

Prueksaritanont, T.

Journal:

Drug Metabolism and Disposition

Année:

2002

Langue:

english

Fichier:

PDF, 356 KB

english, 2002

44

The phenomenon and cause of the dose-dependent oral absorption of chlorothiazide in rats: Extrapolation to human data based on the body surface area concept

Fung-Hwa Hsu, Thomayant Prueksaritanont, Myung G. Lee, Win L. Chiou

Journal:

Journal of Pharmacokinetics and Pharmacodynamics

Année:

1987

Langue:

english

Fichier:

PDF, 1014 KB

english, 1987

45

Effect of P-glycoprotein-mediated efflux on cerebrospinal fluid concentrations in rhesus monkeys

Cuyue Tang, Yuhsin Kuo, Nicole T. Pudvah, Joan D. Ellis, Maria S. Michener, Melissa Egbertson, Samuel L. Graham, Jacquelynn J. Cook, Jerome H. Hochman, Thomayant Prueksaritanont

Journal:

Biochemical Pharmacology

Année:

2009

Langue:

english

Fichier:

PDF, 188 KB

english, 2009

46

Stereospecific reduction of a potent kinesin spindle protein (KSP) inhibitor in human tissues

Chunze Li, Bing Lu, Robert M. Garbaccio, Edward S. Tasber, Mark E. Fraley, George D. Hartman, Jingjing Ye, Jane C. Harrelson, Thomayant Prueksaritanont

Journal:

Biochemical Pharmacology

Année:

2010

Langue:

english

Fichier:

PDF, 516 KB

english, 2010

47

Pharmacokinetics of IgG1 monoclonal antibodies produced in humanized Pichia pastoris with specific glycoforms: A comparative study with CHO produced materials

Liming Liu, Andy Stadheim, Lora Hamuro, Tamara Pittman, Weirong Wang, Dongxing Zha, Jerome Hochman, Thomayant Prueksaritanont

Journal:

Année:

2011

Langue:

english

Fichier:

PDF, 338 KB

english, 2011

48

Impact of methionine oxidation in human IgG1 Fc on serum half-life of monoclonal antibodies

Weirong Wang, Josef Vlasak, Yunsong Li, Pavlo Pristatsky, Yulin Fang, Tamara Pittman, Jeanette Roman, Yang Wang, Thomayant Prueksaritanont, Roxana Ionescu

Journal:

Molecular Immunology

Année:

2011

Langue:

english

Fichier:

PDF, 532 KB

english, 2011

49

Complicating factors in safety testing of drug metabolites: Kinetic differences between generated and preformed metabolites

Thomayant Prueksaritanont, Jiunn H. Lin, Thomas A. Baillie

Journal:

Toxicology and Applied Pharmacology

Année:

2006

Langue:

english

Fichier:

PDF, 200 KB

english, 2006

50

The impact of sialic acids on the pharmacokinetics of a PEGylated erythropoietin

Liming Liu, Huijuan Li, Stephen R. Hamilton, Sujatha Gomathinayagam, William J. Rayfield, Marc van Maanen, Kuo-Chang Yin, Laura Hong, Thomayant Prueksaritanont

Journal:

Journal of Pharmaceutical Sciences

Année:

2012

Langue:

english

Fichier:

PDF, 190 KB

english, 2012